Found 72 recordings
DICL IDIon ChannelCompound FunctionSpeciesValueReferences
DICL_CP_0235961Voltage-gated inwardly rectifying potassium channel KCNH2InhibitorHomo sapiens (Human)Inhibition: 12.82050% inhibition at 1uM10.1371/journal.pone.0199348, 29979714
DICL_CP_0307250Gamma-aminobutyric acid receptor subunit alpha-4/beta-3/deltaActivatorRattus norvegicus (Rat)EC50: 500 nM10.1111/j.1440-1681.2010.05374.x, 20337660
DICL_CP_0314464Gamma-aminobutyric acid receptor subunit alpha-4beta-3/gamma-2sInhibitorRattus norvegicus (Rat)Ki: >10000 nM10.1016/0014-2999(96)00088-x, 8813598
DICL_CP_0314524Gamma-aminobutyric acid receptor subunit alpha-4InhibitorRattus norvegicus (Rat)Ki: 436 nM10.1016/s0028-3908(96)00054-8, 9014146
DICL_CP_0314529Gamma-aminobutyric acid receptor subunit alpha-4beta-3/gamma-2sInhibitorRattus norvegicus (Rat)Ki: 640 nM10.1016/0014-2999(96)00088-x, 8813598
DICL_CP_0316233Gamma-aminobutyric acid receptor subunit alpha-4beta-3/gamma-2sInhibitorRattus norvegicus (Rat)Ki: 693 nM10.1016/0014-2999(96)00088-x, 8813598
DICL_CP_0317968Gamma-aminobutyric acid receptor subunit alpha-4beta-3/gamma-2sInhibitorRattus norvegicus (Rat)Ki: 922 nM10.1016/0014-2999(96)00088-x, 8813598
DICL_CP_0319137Gamma-aminobutyric acid receptor subunit alpha-4InhibitorRattus norvegicus (Rat)Ki: 8 nM10.1016/s0028-3908(96)00054-8, 9014146
DICL_CP_0319139Gamma-aminobutyric acid receptor subunit alpha-4beta-3/gamma-2sInhibitorRattus norvegicus (Rat)Ki: 11.9 nM10.1016/0014-2999(96)00088-x, 8813598
DICL_CP_0320152Gamma-aminobutyric acid receptor subunit alpha-4InhibitorRattus norvegicus (Rat)Ki: 897 nM10.1016/s0028-3908(96)00054-8, 9014146
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